What is Rilmazafone?

Rilmazafone (450191-S) is a water-soluble, open-ring benzodiazepine prodrug, supplied as pressed pellets for laboratory research — each pellet contains 4 mg.

Specifications

• Synonyms: 450191-S, Rhythmy (hydrochloride)
• CAS number: 99593-25-6 (free base); 85815-37-8 (hydrochloride)
• Class: benzodiazepine prodrug (triazolyl aminobenzophenone)
• Molecular formula: C21H20Cl2N6O3
• Molecular weight: ~475.33 g/mol
• Chemical name: 1-[4-chloro-2-(2-chlorobenzoyl)phenyl]-5-[(glycylamino)methyl]-N,N-dimethyl-1H-1,2,4-triazole-3-carboxamide
• Format: pressed pellets · 4 mg per pellet
• Pack sizes: 10 · 25 · 50 pellets
• Storage: keep sealed, cool, dry and away from light

In research settings Rilmazafone is studied as a prodrug that is metabolically converted to rilmazolam, a positive allosteric modulator at the benzodiazepine site of the GABA-A receptor; rilmazafone itself has no intrinsic benzodiazepine-receptor affinity prior to activation.

Limited availability: this is a small one-off batch — stock is restricted while it lasts.

Quality & documentation: every batch is third-party tested; a current Certificate of Analysis is available on request.

Shipping: plain, unbranded packaging shipped from the Netherlands across the EU.

For laboratory research use only. Not for human or veterinary consumption. Buyers must be 18+.